The synthesis of aza-β-lactams via tandem Petasis-Ugi multi-component condensation and 1,3-diisopropylcarbodiimide (DIC) condensation reaction

Published in: Journal, Volume :44, Issue : 33, Pages : 6297-6300

DOI : 10.1016/s0040-4039(03)01524-7

Author : Naskar, Dinabandhu; Roy, Amrita; Seibel, William L.; West, Laura; Portlock, David E.

Abstract : The synthetic utility of a tandem Petasis-Ugi multi-component condensation and 1,3-diisopropylcarbodiimide condensation reactions have been employed to efficiently prepare two to four-dimensional libraries of aza-β-lactams.